PDGs

 

The “druggable genome”, a term coined by Hopkins and Groom in 2002(3), defines a subset of genes in the human genome encoding proteins that may be amenable to modulation by drug-like molecules. To define potentially druggable genes (PDGs) in the human genome, we integrated the PDG candidates generated by six independent studies in which the druggable genes were systematically annotated by different strategies at a whole genome level. .

List of the PDGs in the human genome


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HGNC NameEnsembl Gene IDHGNC SymbolGenomic LocationTDLPubTator Score
taste 2 receptor member 7ENSG00000121377TAS2R7chr12:10801532-10802627:-Tbio3.1
olfactory receptor family 1 subfamily S member 2ENSG00000197887OR1S2chr11:58203202-58204181:-Tdark0
olfactory receptor family 5 subfamily AS member 1ENSG00000181785OR5AS1chr11:56030419-56031393:+Tdark0
olfactory receptor family 4 subfamily F member 15ENSG00000182854OR4F15chr15:101805720-101819147:+Tdark0.166667
olfactory receptor family 8 subfamily K member 1ENSG00000150261OR8K1chr11:56346039-56346998:+Tdark0
olfactory receptor family 5 subfamily B member 21ENSG00000198283OR5B21chr11:58507175-58508105:-Tdark0
olfactory receptor family 5 subfamily AN member 1ENSG00000176495OR5AN1chr11:59364412-59365448:+Tdark1.5
olfactory receptor family 5 subfamily D member 18ENSG00000186119OR5D18chr11:55819630-55820571:+Tdark0
solute carrier family 22 member 24ENSG00000197658SLC22A24chr11:63079940-63144221:-Tdark1.33333
olfactory receptor family 5 subfamily K member 4ENSG00000196098OR5K4chr3:98353854-98354819:+Tdark0
olfactory receptor family 13 subfamily D member 1ENSG00000179055OR13D1chr9:104694422-104695462:+Tdark0
olfactory receptor family 5 subfamily B member 2ENSG00000172365OR5B2chr11:58422265-58423313:-Tdark0
olfactory receptor family 13 subfamily C member 2ENSG00000276119OR13C2chr9:104604671-104605627:-Tdark0
olfactory receptor family 4 subfamily P member 4ENSG00000181927OR4P4chr11:55638358-55639296:+Tdark0.25
olfactory receptor family 8 subfamily G member 1ENSG00000197849OR8G1chr11:124249676-124250611:+Tdark0
olfactory receptor family 9 subfamily G member 4ENSG00000172457OR9G4chr11:56742827-56743811:-Tdark0
olfactory receptor family 4 subfamily C member 13ENSG00000258817OR4C13chr11:49952391-49953419:+Tdark0
olfactory receptor family 6 subfamily C member 68ENSG00000205327OR6C68chr12:55492378-55493316:+Tdark0
olfactory receptor family 13 subfamily F member 1ENSG00000186881OR13F1chr9:104504263-104505222:+Tdark9.33333
olfactory receptor family 9 subfamily A member 2ENSG00000179468OR9A2chr7:143026158-143027195:-Tdark0

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