PDGs
The “druggable genome”, a term coined by Hopkins and Groom in 2002(3), defines a subset of genes in the human genome encoding proteins that may be amenable to modulation by drug-like molecules. To define potentially druggable genes (PDGs) in the human genome, we integrated the PDG candidates generated by six independent studies in which the druggable genes were systematically annotated by different strategies at a whole genome level. .
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| HGNC Name | Ensembl Gene ID | HGNC Symbol | Genomic Location | TDL | PubTator Score |
| serine protease 12 | ENSG00000164099 | PRSS12 | chr4:118280038-118353003:- | Tbio | 12.0876 |
| Fc receptor like 4 | ENSG00000163518 | FCRL4 | chr1:157573749-157598080:- | Tbio | 23.9393 |
| solute carrier family 25 member 12 | ENSG00000115840 | SLC25A12 | chr2:171784370-171999859:- | Tbio | 49.0749 |
| phospholipase A2 group XIIA | ENSG00000123739 | PLA2G12A | chr4:109709989-109730077:- | Tbio | 7.27944 |
| retinoid X receptor beta | ENSG00000204231 | RXRB | chr6:33193588-33200688:- | Tclin | 82.2537 |
| interleukin 9 | ENSG00000145839 | IL9 | chr5:135892246-135895827:- | Tbio | 870.988 |
| ribosomal oxygenase 1 | ENSG00000170468 | C14orf169 | chr14:73490964-73493392:+ | Tbio | 9.61071 |
| solute carrier family 12 member 9 | ENSG00000146828 | SLC12A9 | chr7:100826820-100867009:+ | Tdark | 4.80311 |
| olfactory receptor family 10 subfamily R member 2 | ENSG00000198965 | OR10R2 | chr1:158479878-158480885:+ | Tdark | 220.86 |
| tubulin beta 8B | ENSG00000173213 | TUBB8P12 | chr18:47221-73545:- | Tdark | 0 |
| hydroxysteroid dehydrogenase like 2 | ENSG00000119471 | HSDL2 | chr9:112379937-112472410:+ | Tdark | 3 |
| C-C motif chemokine ligand 3 like 3 | ENSG00000276085 | CCL3L3 | chr17:36194869-36196758:- | 0 | |
| arginyl aminopeptidase like 1 | ENSG00000142327 | RNPEPL1 | chr2:240565804-240581372:+ | Tbio | 1.33333 |
| cripto, FRL-1, cryptic family 1 | ENSG00000136698 | CFC1 | chr2:130592168-130599575:- | Tbio | 810.339 |
| interferon alpha 17 | ENSG00000234829 | IFNA17 | chr9:21206528-21228222:- | Tbio | 220.983 |
| integrator complex subunit 12 | ENSG00000138785 | INTS12 | chr4:105682627-105895986:- | Tbio | 4.78333 |
| CDC42 binding protein kinase beta | ENSG00000198752 | CDC42BPB | chr14:102932379-103057462:- | Tbio | 9.55278 |
| rhomboid like 3 | ENSG00000141314 | RHBDL3 | chr17:32266176-32324661:+ | Tdark | 5.2 |
| myotubularin related protein 1 | ENSG00000063601 | MTMR1 | chrX:150692971-150765103:+ | Tbio | 6.57738 |
| crystallin zeta like 1 | ENSG00000205758 | CRYZL1 | chr21:33589341-33643926:- | Tbio | 2 |
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