PDGs

 

The “druggable genome”, a term coined by Hopkins and Groom in 2002(3), defines a subset of genes in the human genome encoding proteins that may be amenable to modulation by drug-like molecules. To define potentially druggable genes (PDGs) in the human genome, we integrated the PDG candidates generated by six independent studies in which the druggable genes were systematically annotated by different strategies at a whole genome level. .

List of the PDGs in the human genome


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HGNC NameEnsembl Gene IDHGNC SymbolGenomic LocationTDLPubTator Score
phosphoinositide-3-kinase regulatory subunit 6ENSG00000276231PIK3R6chr17:8802723-8867677:-Tbio2.66667
phosphodiesterase 6GENSG00000185527PDE6Gchr17:81650459-81663112:-Tclin8.80556
dehydrogenase/reductase 9ENSG00000073737DHRS9chr2:169064789-169096167:+Tbio11.6635
kelch repeat and BTB domain containing 2ENSG00000170852KBTBD2chr7:32868172-32894131:-Tdark0.2
solute carrier family 28 member 2ENSG00000137860SLC28A2chr15:45252230-45277845:+Tchem56.9575
transient receptor potential cation channel subfamily C member 3ENSG00000138741TRPC3chr4:121879027-121951754:-Tchem208.891
TNF receptor superfamily member 6bENSG00000243509TNFRSF6Bchr20:63696668-63698684:+Tbio169.494
MAPK activated protein kinase 5ENSG00000089022MAPKAPK5chr12:111841978-111902238:+Tchem45.3008
primase and DNA directed polymeraseENSG00000164306PRIMPOLchr4:184649613-184694963:+Tbio21.0833
coenzyme Q6, monooxygenaseENSG00000119723COQ6chr14:73949926-73963670:+Tbio7.28237
SID1 transmembrane family member 2ENSG00000149577SIDT2chr11:117178733-117197445:+Tbio0.375
serine/threonine kinase 38 likeENSG00000211455STK38Lchr12:27243968-27325959:+Tchem8.30516
mannosidase alpha class 2A member 2ENSG00000196547MAN2A2chr15:90902218-90922584:+Tbio2.91667
ATPase H+ transporting V0 subunit a1ENSG00000033627ATP6V0A1chr17:42458844-42522611:+Tbio20.95
TAFA chemokine like family member 4ENSG00000163377FAM19A4chr3:68731766-68932610:-Tbio7.42946
nuclear receptor subfamily 2 group C member 1ENSG00000120798NR2C1chr12:95020229-95073703:-Tbio86.9826
adenosine monophosphate deaminase 1ENSG00000116748AMPD1chr1:114673098-114695618:-Tchem224.867
CD300 molecule like family member gENSG00000161649CD300LGchr17:43847148-43863629:+Tdark5.01786
PWWP domain containing 3A, DNA repair factorENSG00000160953MUM1chr19:1285893-1378431:+Tdark124.54
taste 2 receptor member 19ENSG00000212124TAS2R19chr12:11021619-11022620:-Tdark2.11667

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