PDGs
The “druggable genome”, a term coined by Hopkins and Groom in 2002(3), defines a subset of genes in the human genome encoding proteins that may be amenable to modulation by drug-like molecules. To define potentially druggable genes (PDGs) in the human genome, we integrated the PDG candidates generated by six independent studies in which the druggable genes were systematically annotated by different strategies at a whole genome level. .
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| HGNC Name | Ensembl Gene ID | HGNC Symbol | Genomic Location | TDL | PubTator Score |
| phospholipase A2 group IIF | ENSG00000158786 | PLA2G2F | chr1:20139326-20150386:+ | Tchem | 3.03535 |
| phospholipase C delta 4 | ENSG00000115556 | PLCD4 | chr2:218607765-218637184:+ | Tbio | 12.5012 |
| torsin family 2 member A | ENSG00000160404 | TOR2A | chr9:127731524-127735317:- | Tbio | 12.2833 |
| chloride channel accessory 4 | ENSG00000016602 | CLCA4 | chr1:86547078-86580754:+ | Tbio | 9.93655 |
| solute carrier family 28 member 1 | ENSG00000156222 | SLC28A1 | chr15:84884654-84945796:+ | Tbio | 81.6988 |
| cholinergic receptor nicotinic beta 1 subunit | ENSG00000170175 | CHRNB1 | chr17:7445061-7457707:+ | Tclin | 24.8482 |
| serine peptidase inhibitor Kazal type 13 | ENSG00000214510 | SPINK13 | chr5:148268180-148286254:+ | Tdark | 2.15476 |
| interleukin 12B | ENSG00000113302 | IL12B | chr5:159314783-159330887:- | Tclin | 391.552 |
| cathepsin F | ENSG00000174080 | CTSF | chr11:66563463-66568841:- | Tchem | 27.1873 |
| ubiquitin C-terminal hydrolase L5 | ENSG00000116750 | UCHL5 | chr1:193012250-193060080:- | Tbio | 37.569 |
| leukocyte immunoglobulin like receptor A1 | ENSG00000104974 | LILRA1 | chr19:54573879-54602090:+ | Tdark | 4.33333 |
| pancreatic lipase | ENSG00000175535 | PNLIP | chr10:116545931-116567855:+ | Tclin | 336.767 |
| PDZ domain containing 2 | ENSG00000133401 | PDZD2 | chr5:31639410-32110931:+ | Tbio | 26.6861 |
| histone deacetylase 9 | ENSG00000048052 | HDAC9 | chr7:18086949-19002416:+ | Tclin | 558.949 |
| solute carrier family 8 member A2 | ENSG00000118160 | SLC8A2 | chr19:47428017-47472168:- | Tbio | 24.7286 |
| tubulin beta 6 class V | ENSG00000176014 | TUBB6 | chr18:12307669-12344320:+ | Tclin | 4.99401 |
| gamma-aminobutyric acid type A receptor subunit beta2 | ENSG00000145864 | GABRB2 | chr5:161288429-161549044:- | Tclin | 39.1244 |
| tryptophan hydroxylase 1 | ENSG00000129167 | TPH1 | chr11:18017564-18042426:- | Tclin | 190.041 |
| potassium two pore domain channel subfamily K member 12 | ENSG00000184261 | KCNK12 | chr2:47516581-47570939:- | Tbio | 6.54664 |
| microtubule associated serine/threonine kinase 2 | ENSG00000086015 | MAST2 | chr1:45786987-46036124:+ | Tbio | 20.0247 |
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